Development of an acid ceramidase activity-based probe.

نویسندگان

  • Cécile M J Ouairy
  • Maria J Ferraz
  • Rolf G Boot
  • Marc P Baggelaar
  • Mario van der Stelt
  • Monique Appelman
  • Gijsbert A van der Marel
  • Bogdan I Florea
  • Johannes M F G Aerts
  • Herman S Overkleeft
چکیده

Acid ceramidase is responsible for the ultimate step in the catabolism of (glyco)sphingolipids by hydrolysis of ceramide into sphingosine and free fatty acid. Deficiency in acid ceramidase is the molecular basis of Farber disease. Here we report the synthesis and characterization of an activity-based acid ceramidase probe.

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عنوان ژورنال:
  • Chemical communications

دوره 51 28  شماره 

صفحات  -

تاریخ انتشار 2015